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VRLIVAVRIWRR details
Primary information
ID antitb_1333,
Name23555622
N-Terminal modificationInnate defence regulator peptide 1018
C-Terminal ModificationVRLIVAVRIWRR
Chemical ModificationFree
Linear/CyclicFree
LengthNone
ChiralityLinear
Nature12
SourceL
OriginCationic
SpeciesSynthetic
Inhibition ConcentrationMycobacterium tuberculosis
In Vitro/ In vivoMycobacterium tuberculosis H37Rv
Cell LineMIC = 16.4± 5.4 mg/mL
Inhibition ConcentrationBoth
Sequence2012
CytotoxicityHuman U937 promonocytic cell line
In vivo ModelNA
Lethal DoseNone
Immune ResponceBALB/C
Mechanism of Action32 mg in 100 mL of saline solution (1 mg/kg)
TargetIncrease expression of MCP-1,Gro-α and TNF-α
Combination TherapyNA
Other activitiesNA
PMIDNA
Year of PublicationAntimicrobial against plasmodium aeruginosa/ S. aureus
Tertiary Structure
(Technique)
Not Predicted),